Yang, Xian-Hui

Synthesis, biological evaluation, and molecular docking studies of 1,3,4-thiadiazol-2-amide derivatives as novel anticancer agents. [electronic resource] - Bioorganic & medicinal chemistry May 2012 - 2789-95 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2012.03.040 doi


Amides--chemical synthesis
Antineoplastic Agents--chemical synthesis
Binding Sites
Cell Line, Tumor
Cell Proliferation--drug effects
Computer Simulation
Drug Screening Assays, Antitumor
Focal Adhesion Kinase 1--antagonists & inhibitors
Humans
Protein Kinase Inhibitors--chemical synthesis
Protein Structure, Tertiary
Structure-Activity Relationship
Thiadiazoles--chemistry