Selivanova, Svetlana V

Radiofluorinated histamine H₃ receptor antagonist as a potential probe for in vivo PET imaging: radiosynthesis and pharmacological evaluation. [electronic resource] - Bioorganic & medicinal chemistry May 2012 - 2889-96 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2012.03.024 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Animals
Brain--diagnostic imaging
Cell Line
Dogs
Drug Stability
Fluorine Radioisotopes--chemistry
Histamine H3 Antagonists--chemical synthesis
Humans
Isotope Labeling
Male
Microsomes, Liver--metabolism
Piperidines--chemical synthesis
Positron-Emission Tomography
Protein Binding
Radiopharmaceuticals--chemical synthesis
Rats
Rats, Sprague-Dawley
Receptors, Histamine H3--chemistry