Radiofluorinated histamine H₃ receptor antagonist as a potential probe for in vivo PET imaging: radiosynthesis and pharmacological evaluation. [electronic resource]
- Bioorganic & medicinal chemistry May 2012
- 2889-96 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2012.03.024 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism Animals Brain--diagnostic imaging Cell Line Dogs Drug Stability Fluorine Radioisotopes--chemistry Histamine H3 Antagonists--chemical synthesis Humans Isotope Labeling Male Microsomes, Liver--metabolism Piperidines--chemical synthesis Positron-Emission Tomography Protein Binding Radiopharmaceuticals--chemical synthesis Rats Rats, Sprague-Dawley Receptors, Histamine H3--chemistry