Halestrap, A P

Inhibition of Ca2(+)-induced large-amplitude swelling of liver and heart mitochondria by cyclosporin is probably caused by the inhibitor binding to mitochondrial-matrix peptidyl-prolyl cis-trans isomerase and preventing it interacting with the adenine nucleotide translocase. [electronic resource] - The Biochemical journal May 1990 - 153-60 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0264-6021

10.1042/bj2680153 doi


Adenosine Diphosphate--pharmacology
Amino Acid Isomerases--antagonists & inhibitors
Animals
Bongkrekic Acid--pharmacology
Calcium--pharmacology
Cell Membrane Permeability
Cyclosporins--metabolism
Kinetics
Light
Mitochondria, Heart--drug effects
Mitochondria, Liver--drug effects
Mitochondrial ADP, ATP Translocases--antagonists & inhibitors
Mitochondrial Swelling--drug effects
Nucleotidyltransferases--metabolism
Peptidylprolyl Isomerase
Rats
Scattering, Radiation
Sucrose
Thiocyanates