TY - GEN AU - Dong,Ming-xin AU - Lu,Lu AU - Li,Haitao AU - Wang,Xiaohua AU - Lu,Hong AU - Jiang,Shibo AU - Dai,Qiu-yun TI - Design, synthesis, and biological activity of novel 1,4-disubstituted piperidine/piperazine derivatives as CCR5 antagonist-based HIV-1 entry inhibitors SN - 1464-3405 PY - 2012///1011 KW - Animals KW - Biological Availability KW - CCR5 Receptor Antagonists KW - Cell Line KW - Drug Design KW - HIV Fusion Inhibitors KW - chemical synthesis KW - HIV-1 KW - drug effects KW - Humans KW - Inhibitory Concentration 50 KW - Microbial Sensitivity Tests KW - Piperazines KW - Piperidines KW - Solubility KW - Structure-Activity Relationship N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.bmcl.2012.03.019 ER -