TY  - GEN
AU  - Lebakken,Connie S
AU  - Reichling,Laurie J
AU  - Ellefson,Jason M
AU  - Riddle,Steven M
TI  - Detection of allosteric kinase inhibitors by displacement of active site probes
SN  - 1552-454X
PY  - 2012///0920
KW  - Adenosine Triphosphate
KW  - metabolism
KW  - Allosteric Regulation
KW  - drug effects
KW  - Binding, Competitive
KW  - Catalytic Domain
KW  - Drug Evaluation, Preclinical
KW  - methods
KW  - Fluorescence Resonance Energy Transfer
KW  - Fusion Proteins, bcr-abl
KW  - antagonists & inhibitors
KW  - Humans
KW  - Inhibitory Concentration 50
KW  - MAP Kinase Kinase 1
KW  - Protein Binding
KW  - Protein Kinase Inhibitors
KW  - chemistry
KW  - Protein-Tyrosine Kinases
N1  - Publication Type: Evaluation Study; Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1177/1087057112439889
ER  -