Yin, Shen

Functional selectivity induced by mGlu₄ receptor positive allosteric modulation and concomitant activation of Gq coupled receptors. [electronic resource] - Neuropharmacology Mar 2013 - 122-32 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1873-7064

10.1016/j.neuropharm.2012.03.003 doi


Adenylyl Cyclase Inhibitors
Adenylyl Cyclases--metabolism
Allosteric Regulation--physiology
Animals
Benzopyrans--pharmacology
Calcium--metabolism
Calcium Signaling--drug effects
Cell Line
Excitatory Amino Acid Agonists--pharmacology
Excitatory Amino Acid Antagonists--pharmacology
GTP-Binding Protein alpha Subunits, Gq-G11--physiology
Glutamic Acid--pharmacology
Guinea Pigs
Histamine--pharmacology
Humans
Phosphatidylinositols--metabolism
Rats
Receptors, Histamine H1--physiology
Receptors, Metabotropic Glutamate--agonists
Signal Transduction--drug effects