Keubler, Anja

Drug interaction of efavirenz and midazolam: efavirenz activates the CYP3A-mediated midazolam 1'-hydroxylation in vitro. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Jun 2012 - 1178-82 p. digital

Publication Type: Journal Article

1521-009X

10.1124/dmd.111.043844 doi


Alkynes
Benzoxazines--metabolism
Cyclopropanes
Cytochrome P-450 CYP3A--physiology
Drug Interactions--physiology
Enzyme Activation--drug effects
Humans
Hydroxylation--drug effects
Microsomes, Liver--enzymology
Midazolam--metabolism