Cantin, Louis-David

Discovery of P2X3 selective antagonists for the treatment of chronic pain. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2012 - 2565-71 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2012.01.124 doi


Analgesics--administration & dosage
Animals
Chronic Pain--drug therapy
Dose-Response Relationship, Drug
High-Throughput Screening Assays
Humans
Injections, Spinal
Injections, Subcutaneous
Purinergic P2 Receptor Antagonists--administration & dosage
Pyrimidinones--administration & dosage
Pyrroles--administration & dosage
Rats
Rats, Sprague-Dawley
Receptors, Purinergic P2X3--chemistry
Small Molecule Libraries