Saquinavir inhibits the malaria parasite's chloroquine resistance transporter. [electronic resource]
- Antimicrobial agents and chemotherapy May 2012
- 2283-9 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1098-6596
10.1128/AAC.00166-12 doi
Animals Antimalarials--pharmacology Biological Transport--drug effects Chloroquine--pharmacology Drug Combinations Drug Synergism Female HIV Protease Inhibitors--pharmacology Humans Lopinavir--pharmacology Malaria, Falciparum--drug therapy Membrane Transport Proteins--genetics Mutation Oocytes--cytology Plasmodium falciparum--drug effects Protozoan Proteins--antagonists & inhibitors Ritonavir--pharmacology Saquinavir--pharmacology Tritium Xenopus laevis