Investigating the kinetic mechanism of inhibition of elongation factor 2 kinase by NH125: evidence of a common in vitro artifact. [electronic resource]
- Biochemistry Mar 2012
- 2100-12 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4995
10.1021/bi201787p doi
Adenosine Triphosphate--metabolism Amino Acid Sequence Artifacts Cell Line Dose-Response Relationship, Drug Elongation Factor 2 Kinase--antagonists & inhibitors HEK293 Cells Humans Imidazoles--administration & dosage In Vitro Techniques Kinetics Molecular Sequence Data Peptides--chemistry Phosphorylation Protein Kinase Inhibitors--administration & dosage Recombinant Proteins--antagonists & inhibitors Substrate Specificity