TY - GEN AU - Ehmke,Veronika AU - Quinsaat,Jose Enrico Q AU - Rivera-Fuentes,Pablo AU - Heindl,Cornelia AU - Freymond,Céline AU - Rottmann,Matthias AU - Brun,Reto AU - Schirmeister,Tanja AU - Diederich,François TI - Tuning and predicting biological affinity: aryl nitriles as cysteine protease inhibitors SN - 1477-0539 PY - 2012///1119 KW - Catalytic Domain KW - Cathepsin L KW - antagonists & inhibitors KW - Cysteine Endopeptidases KW - chemistry KW - Cysteine Proteinase Inhibitors KW - chemical synthesis KW - Drug Design KW - Humans KW - Models, Molecular KW - Nitriles KW - Trypanosoma brucei brucei KW - enzymology N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1039/c2ob00034b ER -