Use of the cassette-dosing approach to assess brain penetration in drug discovery. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals May 2012
- 963-9 p. digital
Publication Type: Journal Article
1521-009X
10.1124/dmd.111.044420 doi
ATP Binding Cassette Transporter, Subfamily B--genetics ATP Binding Cassette Transporter, Subfamily G, Member 2 ATP-Binding Cassette Transporters--genetics Animals Biological Transport Brain--metabolism Chromatography, High Pressure Liquid Dose-Response Relationship, Drug Drug Discovery--methods Drug Interactions Injections, Subcutaneous Limit of Detection Mice Mice, Knockout Models, Biological Pharmaceutical Preparations--administration & dosage Substrate Specificity Tandem Mass Spectrometry ATP-Binding Cassette Sub-Family B Member 4