Caboni, Laura <br/><br/>
"True" antiandrogens-selective non-ligand-binding pocket disruptors of androgen receptor-coactivator interactions: novel tools for prostate cancer.  [electronic resource] 

 -  Journal of medicinal chemistry  Feb 2012 
 - 1635-44 p.  digital 
<br/><br/> Publication Type: Journal Article; Research Support, Non-U.S. Gov't 
<br/><br/><label>ISSN: </label>1520-4804 
<br/><br/><label>Standard No.: </label>10.1021/jm201438f  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Androgen Antagonists--chemical synthesis<br/>Antineoplastic Agents--chemical synthesis<br/>Cell Proliferation--drug effects<br/>Cell Survival--drug effects<br/>Databases, Factual<br/>Drug Screening Assays, Antitumor<br/>Estrogen Receptor alpha--metabolism<br/>Estrogen Receptor beta--metabolism<br/>Fluorescence Polarization<br/>Fluorescence Resonance Energy Transfer<br/>Humans<br/>Hydrazines--chemical synthesis<br/>Male<br/>Models, Molecular<br/>Nuclear Receptor Coactivators--metabolism<br/>Prostate-Specific Antigen--metabolism<br/>Prostatic Neoplasms--drug therapy<br/>Receptors, Androgen--metabolism<br/>Receptors, Glucocorticoid--metabolism<br/>Receptors, Progesterone--antagonists & inhibitors<br/>Structure-Activity Relationship