Impact of CYP3A5 and ABCB1 gene polymorphisms on fentanyl pharmacokinetics and clinical responses in cancer patients undergoing conversion to a transdermal system. [electronic resource]
- Drug metabolism and pharmacokinetics 2012
- 414-21 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1880-0920
10.2133/dmpk.dmpk-11-rg-134 doi
ATP Binding Cassette Transporter, Subfamily B ATP Binding Cassette Transporter, Subfamily B, Member 1--genetics Administration, Cutaneous Aged Analgesics, Opioid--administration & dosage Cytochrome P-450 CYP3A--genetics Drug Monitoring Female Fentanyl--administration & dosage Genotype Humans Japan Logistic Models Male Middle Aged Neoplasms--drug therapy Odds Ratio Pharmacogenetics Phenotype Polymorphism, Genetic