Characterization of suramin binding sites on the human group IIA secreted phospholipase A2 by site-directed mutagenesis and molecular dynamics simulation. [electronic resource]
- Archives of biochemistry and biophysics Mar 2012
- 17-22 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1096-0384
10.1016/j.abb.2012.01.002 doi
Binding Sites Fluoresceins--chemistry Group II Phospholipases A2--antagonists & inhibitors Humans Hydrophobic and Hydrophilic Interactions Liposomes--chemistry Models, Molecular Molecular Dynamics Simulation Mutagenesis, Site-Directed Protein Binding Protein Conformation Recombinant Proteins--antagonists & inhibitors Spectrometry, Fluorescence Static Electricity Structure-Activity Relationship Suramin--chemistry