Zhou, Wen-jing

Crizotinib (PF-02341066) reverses multidrug resistance in cancer cells by inhibiting the function of P-glycoprotein. [electronic resource] - British journal of pharmacology Jul 2012 - 1669-83 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1476-5381

10.1111/j.1476-5381.2012.01849.x doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Adenosine Triphosphatases--metabolism
Animals
Antineoplastic Agents--pharmacology
Cell Line, Tumor
Crizotinib
Doxorubicin--pharmacokinetics
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Female
Humans
Mice
Mice, Nude
Neoplasms--drug therapy
Paclitaxel--therapeutic use
Protein Kinase Inhibitors--pharmacology
Pyrazoles--pharmacology
Pyridines--pharmacology
Rhodamine 123--pharmacokinetics
Tumor Burden--drug effects
Xenograft Model Antitumor Assays