Gupta, Pankaj

Lack of effect of tofacitinib (CP-690,550) on the pharmacokinetics of the CYP3A4 substrate midazolam in healthy volunteers: confirmation of in vitro data. [electronic resource] - British journal of clinical pharmacology Jul 2012 - 109-15 p. digital

Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't

1365-2125

10.1111/j.1365-2125.2012.04168.x doi


Adult
Cross-Over Studies
Cytochrome P-450 CYP3A--metabolism
Drug Interactions
Female
GABA Modulators--pharmacokinetics
Half-Life
Humans
Janus Kinases--antagonists & inhibitors
Male
Metabolic Clearance Rate
Midazolam--pharmacokinetics
Middle Aged
Piperidines
Pyrimidines--pharmacology
Pyrroles--pharmacology
Young Adult