Tarcsay, Akos

Impact of lipophilic efficiency on compound quality. [electronic resource] - Journal of medicinal chemistry Feb 2012 - 1252-60 p. digital

Publication Type: Journal Article

1520-4804

10.1021/jm201388p doi


Biological Transport, Active
Central Nervous System Agents--adverse effects
Chemistry, Physical
Drug Discovery
Drug-Related Side Effects and Adverse Reactions
Microsomes--metabolism
Octanols
Permeability
Pharmaceutical Preparations--chemistry
Protein Binding
Structure-Activity Relationship
Thermodynamics
Water