Impact of lipophilic efficiency on compound quality. [electronic resource]
- Journal of medicinal chemistry Feb 2012
- 1252-60 p. digital
Publication Type: Journal Article
1520-4804
10.1021/jm201388p doi
Biological Transport, Active Central Nervous System Agents--adverse effects Chemistry, Physical Drug Discovery Drug-Related Side Effects and Adverse Reactions Microsomes--metabolism Octanols Permeability Pharmaceutical Preparations--chemistry Protein Binding Structure-Activity Relationship Thermodynamics Water