Tian, Wang
Structure-based discovery of a novel inhibitor targeting the β-catenin/Tcf4 interaction. [electronic resource]
- Biochemistry Jan 2012
- 724-31 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
ISSN: 1520-4995
Standard No.: 10.1021/bi201428h doi
Subjects--Topical Terms: Antineoplastic Agents--pharmacology Basic Helix-Loop-Helix Leucine Zipper Transcription Factors--chemistry Basic Helix-Loop-Helix Transcription Factors--metabolism Cell Proliferation--drug effects Cell Survival--drug effects Crystallography, X-Ray Down-Regulation--drug effects Drug Evaluation, Preclinical--methods HCT116 Cells Humans Models, Molecular Protein Binding--drug effects Protein Conformation Small Molecule Libraries--pharmacology Transcription Factor 4 Transcription Factors--chemistry Transcription, Genetic--drug effects User-Computer Interface Wnt Signaling Pathway--drug effects beta Catenin--chemistry