Tian, Wang

Structure-based discovery of a novel inhibitor targeting the β-catenin/Tcf4 interaction. [electronic resource] - Biochemistry Jan 2012 - 724-31 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4995

10.1021/bi201428h doi


Antineoplastic Agents--pharmacology
Basic Helix-Loop-Helix Leucine Zipper Transcription Factors--chemistry
Basic Helix-Loop-Helix Transcription Factors--metabolism
Cell Proliferation--drug effects
Cell Survival--drug effects
Crystallography, X-Ray
Down-Regulation--drug effects
Drug Evaluation, Preclinical--methods
HCT116 Cells
Humans
Models, Molecular
Protein Binding--drug effects
Protein Conformation
Small Molecule Libraries--pharmacology
Transcription Factor 4
Transcription Factors--chemistry
Transcription, Genetic--drug effects
User-Computer Interface
Wnt Signaling Pathway--drug effects
beta Catenin--chemistry