Bali, Ustav Design and synthesis of potent carboxylic acid DGAT1 inhibitors with high cell permeability. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2012 - 824-8 p. digital Publication Type: Journal Article ISSN: 1464-3405 Standard No.: 10.1016/j.bmcl.2011.12.050 doi Subjects--Topical Terms: Caco-2 CellsDiacylglycerol O-Acyltransferase--antagonists & inhibitorsDose-Response Relationship, DrugDrug DesignEnzyme Inhibitors--chemical synthesisHumansMolecular StructurePermeability--drug effectsStructure-Activity Relationship