Montano, Ryan

Preclinical development of the novel Chk1 inhibitor SCH900776 in combination with DNA-damaging agents and antimetabolites. [electronic resource] - Molecular cancer therapeutics Feb 2012 - 427-38 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1538-8514

10.1158/1535-7163.MCT-11-0406 doi


Antimetabolites--pharmacology
Antineoplastic Agents--pharmacology
Blotting, Western
Camptothecin--analogs & derivatives
Cell Cycle Checkpoints--drug effects
Cell Line
Cell Line, Tumor
Cell Proliferation--drug effects
Cell Survival--drug effects
Checkpoint Kinase 1
Cytarabine--pharmacology
DNA Breaks, Double-Stranded--drug effects
DNA Damage
Deoxycytidine--analogs & derivatives
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Drug Synergism
Flow Cytometry
Humans
Hydroxyurea--pharmacology
Irinotecan
Molecular Structure
Phosphorylation--drug effects
Protein Kinase Inhibitors--chemistry
Protein Kinases--metabolism
Pyrazoles--chemistry
Pyrimidines--chemistry
Staurosporine--analogs & derivatives
Gemcitabine