TY - GEN AU - Ito,Shinji AU - Terasaka,Tadashi AU - Zenkoh,Tatsuya AU - Matsuda,Hiroshi AU - Hayashida,Hisashi AU - Nagata,Hiroshi AU - Imamura,Yoshimasa AU - Kobayashi,Miki AU - Takeuchi,Makoto AU - Ohta,Mitsuaki TI - Discovery of novel and potent CRTH2 antagonists SN - 1464-3405 PY - 2012///0824 KW - Administration, Oral KW - Animals KW - Biological Availability KW - Dose-Response Relationship, Drug KW - Drug Discovery KW - Guinea Pigs KW - HEK293 Cells KW - Humans KW - Molecular Structure KW - Receptors, Immunologic KW - antagonists & inhibitors KW - Receptors, Prostaglandin KW - Stereoisomerism KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2011.11.079 ER -