Melancon, Bruce J

Allosteric modulation of seven transmembrane spanning receptors: theory, practice, and opportunities for central nervous system drug discovery. [electronic resource] - Journal of medicinal chemistry Feb 2012 - 1445-64 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1520-4804

10.1021/jm201139r doi


Allosteric Regulation
Animals
Central Nervous System Agents--chemistry
Drug Discovery
Humans
Ligands
Receptors, G-Protein-Coupled--agonists
Receptors, Metabotropic Glutamate--metabolism
Receptors, Muscarinic--metabolism
Structure-Activity Relationship