Modification of HIV-1 reverse transcriptase and integrase activity by gold(III) complexes in direct biochemical assays. [electronic resource]
- Bioorganic & medicinal chemistry Jan 2012
- 401-7 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2011.10.072 doi
Binding Sites Computer Simulation Coordination Complexes--chemistry Gold--chemistry HIV Integrase--chemistry HIV Integrase Inhibitors--chemical synthesis HIV Reverse Transcriptase--antagonists & inhibitors HIV-1--drug effects Humans Leukocytes, Mononuclear--drug effects Reverse Transcriptase Inhibitors--chemical synthesis