YHHU0895, a novel synthetic small-molecule microtubule-destabilizing agent, effectively overcomes P-glycoprotein-mediated tumor multidrug resistance. [electronic resource]
- Cancer letters Jan 2012
- 54-62 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1872-7980
10.1016/j.canlet.2011.09.013 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--physiology Animals Antineoplastic Agents--pharmacology Cell Line, Tumor Drug Resistance, Multiple Drug Resistance, Neoplasm Female Humans Indoles--pharmacology Mice Microtubules--drug effects Polymerization Pyrimidines--pharmacology Tubulin--metabolism Xenograft Model Antitumor Assays