TY  - GEN
AU  - Mitch,Charles H
AU  - Quimby,Steven J
AU  - Diaz,Nuria
AU  - Pedregal,Concepcion
AU  - de la Torre,Marta G
AU  - Jimenez,Alma
AU  - Shi,Qing
AU  - Canada,Emily J
AU  - Kahl,Steven D
AU  - Statnick,Michael A
AU  - McKinzie,David L
AU  - Benesh,Dana R
AU  - Rash,Karen S
AU  - Barth,Vanessa N
TI  - Discovery of aminobenzyloxyarylamides as κ opioid receptor selective antagonists: application to preclinical development of a κ opioid receptor antagonist receptor occupancy tracer
SN  - 1520-4804
PY  - 2012///0305
KW  - Animals
KW  - Benzamides
KW  - chemical synthesis
KW  - Brain
KW  - metabolism
KW  - CHO Cells
KW  - Chromatography, Liquid
KW  - Cricetinae
KW  - Cricetulus
KW  - HEK293 Cells
KW  - Humans
KW  - Pyrrolidines
KW  - Radioligand Assay
KW  - Rats
KW  - Receptors, Opioid, kappa
KW  - antagonists & inhibitors
KW  - Stereoisomerism
KW  - Structure-Activity Relationship
KW  - Tandem Mass Spectrometry
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1021/jm200789r
ER  -