TY - GEN AU - Barnes,Matthew J AU - Burschka,Christian AU - Büttner,Matthias W AU - Conroy,Richard AU - Daiss,Jürgen O AU - Gray,Ian C AU - Hendrick,Alan G AU - Tam,L H AU - Kuehn,Diana AU - Miller,David J AU - Mills,John S AU - Mitchell,Philip AU - Montana,John G AU - Muniandy,Parameswary A AU - Rapley,Helen AU - Showell,Graham A AU - Tebbe,David AU - Tacke,Reinhold AU - Warneck,Julie B H AU - Zhu,Bin TI - Silicon analogues of the nonpeptidic GnRH antagonist AG-045572: syntheses, crystal structure analyses, and pharmacological characterization SN - 1860-7187 PY - 2012///0413 KW - Animals KW - Crystallography, X-Ray KW - Drug Evaluation, Preclinical KW - Furans KW - chemistry KW - Gonadotropin-Releasing Hormone KW - antagonists & inhibitors KW - Hormone Antagonists KW - Humans KW - Luteinizing Hormone KW - Magnetic Resonance Spectroscopy KW - Male KW - Molecular Structure KW - Orchiectomy KW - Rats, Wistar KW - Receptors, LHRH KW - genetics KW - Silicon KW - Structure-Activity Relationship KW - Tetrahydronaphthalenes N1 - Publication Type: Journal Article UR - https://doi.org/10.1002/cmdc.201100318 ER -