TY - GEN AU - Wempe,Michael F AU - Rice,Peter J AU - Lightner,Janet W AU - Jutabha,Promsuk AU - Hayashi,Michinari AU - Anzai,Naohiko AU - Wakui,Shin AU - Kusuhara,Hiroyuki AU - Sugiyama,Yuichi AU - Endou,Hitoshi TI - Metabolism and pharmacokinetic studies of JPH203, an L-amino acid transporter 1 (LAT1) selective compound SN - 1880-0920 PY - 2012///0716 KW - Acetylation KW - Animals KW - Antineoplastic Agents KW - analysis KW - Benzoxazoles KW - Biotransformation KW - Dogs KW - Humans KW - Intestine, Small KW - metabolism KW - Kidney KW - chemistry KW - Large Neutral Amino Acid-Transporter 1 KW - Liver KW - Macaca fascicularis KW - Male KW - Membrane Transport Modulators KW - Mice KW - Microsomes KW - Microsomes, Liver KW - Rats KW - Rats, Sprague-Dawley KW - Tissue Distribution KW - Tyrosine KW - analogs & derivatives N1 - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't UR - https://doi.org/10.2133/dmpk.dmpk-11-rg-091 ER -