Metabolism and pharmacokinetic studies of JPH203, an L-amino acid transporter 1 (LAT1) selective compound. [electronic resource]
- Drug metabolism and pharmacokinetics 2012
- 155-61 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1880-0920
10.2133/dmpk.dmpk-11-rg-091 doi
Acetylation Animals Antineoplastic Agents--analysis Benzoxazoles--analysis Biotransformation Dogs Humans Intestine, Small--metabolism Kidney--chemistry Large Neutral Amino Acid-Transporter 1--chemistry Liver--chemistry Macaca fascicularis Male Membrane Transport Modulators--analysis Mice Microsomes--metabolism Microsomes, Liver--metabolism Rats Rats, Sprague-Dawley Tissue Distribution Tyrosine--analogs & derivatives