Biochemistry and biology of 2'-Fluoro-2'-deoxythymidine (FT), a putative highly selective substrate for thymidine kinase type 2 (TK2). [electronic resource]
- Current radiopharmaceuticals Jan 2012
- 38-46 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1874-4729
10.2174/1874471011205010038 doi
Animals Antineoplastic Agents--pharmacology Autoradiography Bone Neoplasms--drug therapy Cell Line, Tumor Dose-Response Relationship, Drug Drug Screening Assays, Antitumor Humans Inhibitory Concentration 50 Membrane Transport Proteins--metabolism Mice Mice, Inbred BALB C Neoplasm Transplantation Osteosarcoma--drug therapy Phosphorylation Positron-Emission Tomography Radiopharmaceuticals Thymidine--analogs & derivatives Thymidine Kinase Transgenes