Karonen, Tiina

CYP2C8 but not CYP3A4 is important in the pharmacokinetics of montelukast. [electronic resource] - British journal of clinical pharmacology Feb 2012 - 257-67 p. digital

Publication Type: Clinical Trial, Phase IV; Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't

1365-2125

10.1111/j.1365-2125.2011.04086.x doi


14-alpha Demethylase Inhibitors--pharmacology
Acetates--pharmacokinetics
Adult
Anti-Asthmatic Agents--pharmacokinetics
Area Under Curve
Aryl Hydrocarbon Hydroxylases--physiology
Cross-Over Studies
Cyclopropanes
Cytochrome P-450 CYP2C8
Cytochrome P-450 CYP3A--physiology
Drug Interactions
Female
Gemfibrozil--pharmacology
Humans
Hypolipidemic Agents--pharmacology
Itraconazole--pharmacology
Male
Quinolines--pharmacokinetics
Sulfides
Young Adult