High-throughput kinase profiling: a more efficient approach toward the discovery of new kinase inhibitors. [electronic resource]
- Chemistry & biology Jul 2011
- 868-79 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1879-1301
10.1016/j.chembiol.2011.05.010 doi
Aurora Kinases Benzodiazepines--chemistry Drug Evaluation, Preclinical--methods Furans--chemistry High-Throughput Screening Assays--methods Humans Mitogen-Activated Protein Kinase 7--antagonists & inhibitors Models, Molecular Protein Kinase Inhibitors--chemistry Protein Kinases--metabolism Protein Serine-Threonine Kinases--antagonists & inhibitors Protein-Tyrosine Kinases--antagonists & inhibitors Proto-Oncogene Proteins c-pim-1--antagonists & inhibitors Thiazolidinediones--chemistry