TY  - GEN
AU  - Sime,Mairi
AU  - Allan,Amanda C
AU  - Chapman,Paul
AU  - Fieldhouse,Charlotte
AU  - Giblin,Gerard M P
AU  - Healy,Mark P
AU  - Lambert,Millard H
AU  - Leesnitzer,Lisa M
AU  - Lewis,Ann
AU  - Merrihew,Raymond V
AU  - Rutter,Richard A
AU  - Sasse,Rosemary
AU  - Shearer,Barry G
AU  - Willson,Timothy M
AU  - Wilson,Timothy M
AU  - Xu,Robert X
AU  - Virley,David J
TI  - Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARγ partial agonist
SN  - 1464-3405
PY  - 2011///1219
KW  - Benzimidazoles
KW  - chemical synthesis
KW  - Dose-Response Relationship, Drug
KW  - Drug Discovery
KW  - Molecular Structure
KW  - PPAR gamma
KW  - antagonists & inhibitors
KW  - Stereoisomerism
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1016/j.bmcl.2011.06.088
ER  -