Sime, Mairi
Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARγ partial agonist. [electronic resource]
- Bioorganic & medicinal chemistry letters Sep 2011
- 5568-72 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2011.06.088 doi
Benzimidazoles--chemical synthesis
Dose-Response Relationship, Drug
Drug Discovery
Molecular Structure
PPAR gamma--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship