Sime, Mairi

Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARγ partial agonist. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2011 - 5568-72 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2011.06.088 doi


Benzimidazoles--chemical synthesis
Dose-Response Relationship, Drug
Drug Discovery
Molecular Structure
PPAR gamma--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship