Hu, Yonghan

Discovery of indazoles as inhibitors of Tpl2 kinase. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2011 - 4758-61 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2011.06.065 doi


Dose-Response Relationship, Drug
Drug Discovery
Enzyme Inhibitors--chemical synthesis
Humans
Indazoles--chemical synthesis
MAP Kinase Kinase Kinases--antagonists & inhibitors
Models, Molecular
Molecular Structure
Monocytes--enzymology
Proto-Oncogene Proteins--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship