Hu, Yonghan
Discovery of indazoles as inhibitors of Tpl2 kinase. [electronic resource]
- Bioorganic & medicinal chemistry letters Aug 2011
- 4758-61 p. digital
Publication Type: Journal Article
1464-3405
10.1016/j.bmcl.2011.06.065 doi
Dose-Response Relationship, Drug
Drug Discovery
Enzyme Inhibitors--chemical synthesis
Humans
Indazoles--chemical synthesis
MAP Kinase Kinase Kinases--antagonists & inhibitors
Models, Molecular
Molecular Structure
Monocytes--enzymology
Proto-Oncogene Proteins--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship