Sielaff, Frank
Development of substrate analogue inhibitors for the human airway trypsin-like protease HAT. [electronic resource]
- Bioorganic & medicinal chemistry letters Aug 2011
- 4860-4 p. digital
Publication Type: Journal Article
ISSN: 1464-3405
Standard No.: 10.1016/j.bmcl.2011.06.033 doi
Subjects--Topical Terms: Amidines--chemical synthesis Antiviral Agents--chemical synthesis Benzyl Compounds--chemical synthesis Cells, Cultured Dipeptides--chemical synthesis Dose-Response Relationship, Drug Humans Microbial Sensitivity Tests Molecular Structure Orthomyxoviridae--drug effects Serine Endopeptidases--metabolism Serine Proteinase Inhibitors--chemical synthesis Stereoisomerism Structure-Activity Relationship Substrate Specificity Virus Replication--drug effects