Sielaff, Frank

Development of substrate analogue inhibitors for the human airway trypsin-like protease HAT. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2011 - 4860-4 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2011.06.033 doi


Amidines--chemical synthesis
Antiviral Agents--chemical synthesis
Benzyl Compounds--chemical synthesis
Cells, Cultured
Dipeptides--chemical synthesis
Dose-Response Relationship, Drug
Humans
Microbial Sensitivity Tests
Molecular Structure
Orthomyxoviridae--drug effects
Serine Endopeptidases--metabolism
Serine Proteinase Inhibitors--chemical synthesis
Stereoisomerism
Structure-Activity Relationship
Substrate Specificity
Virus Replication--drug effects