Azuma, Junichi

The relationship between clinical pharmacokinetics of aripiprazole and CYP2D6 genetic polymorphism: effects of CYP enzyme inhibition by coadministration of paroxetine or fluvoxamine. [electronic resource] - European journal of clinical pharmacology Jan 2012 - 29-37 p. digital

Publication Type: Comparative Study; Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't

1432-1041

10.1007/s00228-011-1094-4 doi


Adult
Antipsychotic Agents--adverse effects
Aripiprazole
Biotransformation
Cytochrome P-450 CYP2D6--genetics
Cytochrome P-450 CYP2D6 Inhibitors
Cytochrome P-450 CYP3A
Cytochrome P-450 CYP3A Inhibitors
Drug Interactions
Enzyme Inhibitors--adverse effects
Fluvoxamine--adverse effects
Genetic Association Studies
Half-Life
Humans
Japan
Male
Metabolic Clearance Rate--drug effects
Paroxetine--adverse effects
Piperazines--adverse effects
Polymorphism, Genetic
Quinolones--adverse effects
Serotonin 5-HT2 Receptor Antagonists--adverse effects
Selective Serotonin Reuptake Inhibitors--adverse effects
Young Adult