TY  - GEN
AU  - Kerns,Jeffrey K
AU  - Nie,Hong
AU  - Bondinell,William
AU  - Widdowson,Katherine L
AU  - Yamashita,Dennis S
AU  - Rahman,Attiq
AU  - Podolin,Patricia L
AU  - Carpenter,Donald C
AU  - Jin,Qi
AU  - Riflade,Benoit
AU  - Dong,Xiaoyang
AU  - Nevins,Neysa
AU  - Keller,Paul M
AU  - Mitchell,Laura
AU  - Tomaszek,Thaddeus
TI  - Azepanone-based inhibitors of human cathepsin S: optimization of selectivity via the P2 substituent
SN  - 1464-3405
PY  - 2011///1122
KW  - Alanine
KW  - chemistry
KW  - Azepines
KW  - chemical synthesis
KW  - Binding Sites
KW  - Cathepsin K
KW  - antagonists & inhibitors
KW  - Cathepsin L
KW  - Cathepsins
KW  - Computer Simulation
KW  - Humans
KW  - Niacinamide
KW  - analogs & derivatives
KW  - Protease Inhibitors
KW  - Stereoisomerism
KW  - Structure-Activity Relationship
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1016/j.bmcl.2011.06.045
ER  -