Ruschak, Amy M Novel proteasome inhibitors to overcome bortezomib resistance. [electronic resource] - Journal of the National Cancer Institute Jul 2011 - 1007-17 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Review ISSN: 1460-2105 Standard No.: 10.1093/jnci/djr160 doi Subjects--Topical Terms: Allosteric Site--drug effectsAnimalsAntineoplastic Agents--pharmacologyApoptosis--drug effectsBoronic Acids--pharmacologyBortezomibCell Line, TumorChloroquine--pharmacologyClioquinol--pharmacologyDrug Resistance, Neoplasm--drug effectsHumansHydroxyquinolines--pharmacologyLactones--pharmacologyNeoplasms--drug therapyOligopeptides--pharmacologyProtease Inhibitors--pharmacologyProteasome Endopeptidase Complex--chemistryProteasome InhibitorsPyrazines--pharmacologyPyrroles--pharmacologyThreonine--analogs & derivativesUbiquitinated Proteins--metabolismUbiquitination--drug effects