Discovery of orally active, potent, and selective benzotriazole-based PTP1B inhibitors. [electronic resource]
- ChemMedChem Jun 2011
- 1011-6 p. digital
Publication Type: Journal Article
1860-7187
10.1002/cmdc.201100077 doi
Administration, Oral Animals Diabetes Mellitus--drug therapy Enzyme Inhibitors--chemistry Humans Hypoglycemic Agents--chemistry Male Mice Mice, Inbred C57BL Models, Molecular Protein Binding Protein Tyrosine Phosphatase, Non-Receptor Type 1--antagonists & inhibitors Rats Rats, Wistar Structure-Activity Relationship Triazoles--chemistry