Potent and selective phosphopeptide mimetic prodrugs targeted to the Src homology 2 (SH2) domain of signal transducer and activator of transcription 3. [electronic resource]
- Journal of medicinal chemistry May 2011
- 3549-63 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4804
10.1021/jm2000882 doi
Active Transport, Cell Nucleus Antineoplastic Agents--pharmacology Cell Line, Tumor Chemistry, Pharmaceutical--methods Drug Design Drug Screening Assays, Antitumor Humans Kinetics Models, Chemical Phosphatidylinositol 3-Kinases--metabolism Phosphorylation Prodrugs Protein Structure, Tertiary STAT3 Transcription Factor--chemistry Signal Transduction src Homology Domains