Kubota, Katsumi Synthesis and structure-activity relationship of tricyclic carboxylic acids as novel anti-histamines. [electronic resource] - Bioorganic & medicinal chemistry May 2011 - 3005-21 p. digital Publication Type: Journal Article ISSN: 1464-3391 Standard No.: 10.1016/j.bmc.2011.03.003 doi Subjects--Topical Terms: AnimalsAnti-Inflammatory Agents--chemical synthesisAzepines--chemical synthesisCaco-2 CellsCarboxylic Acids--chemical synthesisCell Membrane PermeabilityCyclizationHistamine H1 Antagonists--chemical synthesisHumansMiceOxazepines--chemical synthesisProtein BindingPyrimidines--chemical synthesisRatsReceptors, Histamine H1--chemistryStructure-Activity Relationship