Yao, Zhangyu

Preparation and evaluation of tetrabenazine enantiomers and all eight stereoisomers of dihydrotetrabenazine as VMAT2 inhibitors. [electronic resource] - European journal of medicinal chemistry May 2011 - 1841-8 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't

1768-3254

10.1016/j.ejmech.2011.02.046 doi


Animals
Male
Molecular Conformation
Rats
Rats, Sprague-Dawley
Stereoisomerism
Structure-Activity Relationship
Tetrabenazine--analogs & derivatives
Vesicular Monoamine Transport Proteins--antagonists & inhibitors