Preparation and evaluation of tetrabenazine enantiomers and all eight stereoisomers of dihydrotetrabenazine as VMAT2 inhibitors. [electronic resource]
- European journal of medicinal chemistry May 2011
- 1841-8 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't
1768-3254
10.1016/j.ejmech.2011.02.046 doi
Animals Male Molecular Conformation Rats Rats, Sprague-Dawley Stereoisomerism Structure-Activity Relationship Tetrabenazine--analogs & derivatives Vesicular Monoamine Transport Proteins--antagonists & inhibitors