Structural simplification of bioactive natural products with multicomponent synthesis. 3. Fused uracil-containing heterocycles as novel topoisomerase-targeting agents. [electronic resource]
- Journal of medicinal chemistry Apr 2011
- 2012-21 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1520-4804
10.1021/jm1009428 doi
Antineoplastic Agents--chemical synthesis Biological Products--chemical synthesis Cell Line, Tumor Cell Proliferation--drug effects DNA Topoisomerases, Type I--metabolism DNA Topoisomerases, Type II--metabolism Humans Inhibitory Concentration 50 Topoisomerase II Inhibitors--chemical synthesis Uracil--chemical synthesis