Sedlák, David

Two panels of steroid receptor luciferase reporter cell lines for compound profiling. [electronic resource] - Combinatorial chemistry & high throughput screening May 2011 - 248-66 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1875-5402

10.2174/138620711795222446 doi


Cell Line, Tumor
Dose-Response Relationship, Drug
Drug Discovery--methods
Genes, Reporter
Genetic Engineering--methods
High-Throughput Screening Assays--methods
Humans
Luciferases--genetics
Plasmids--genetics
Promoter Regions, Genetic--drug effects
Receptors, Steroid--agonists
Recombinant Proteins--genetics
Sequence Deletion
Small Molecule Libraries--analysis
Steroids--pharmacology
Transcription Factors--genetics
Transcriptional Activation--drug effects
Transfection