Next-generation Akt inhibitors provide greater specificity: effects on glucose metabolism in adipocytes. [electronic resource]
- The Biochemical journal Apr 2011
- 539-44 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1470-8728
10.1042/BJ20110040 doi
3T3-L1 Cells Adipocytes--drug effects Animals Antineoplastic Agents--pharmacology Cells, Cultured Dose-Response Relationship, Drug Drug Evaluation, Preclinical Glucose--metabolism Glucose Transporter Type 4--metabolism Heterocyclic Compounds, 3-Ring--pharmacology Humans Mice Protein Kinase Inhibitors--pharmacology Protein Transport--drug effects Proto-Oncogene Proteins c-akt--antagonists & inhibitors Substrate Specificity--drug effects