Majmudar, Jaimeen D

Probing the isoprenylcysteine carboxyl methyltransferase (Icmt) binding pocket: sulfonamide modified farnesyl cysteine (SMFC) analogs as Icmt inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters May 2011 - 2616-20 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1464-3405

10.1016/j.bmcl.2011.01.078 doi


Binding Sites
Cysteine--analogs & derivatives
Enzyme Activation--drug effects
Enzyme Inhibitors--chemistry
Humans
Inhibitory Concentration 50
Molecular Structure
Protein Methyltransferases--antagonists & inhibitors
Protein Processing, Post-Translational