Majmudar, Jaimeen D
Probing the isoprenylcysteine carboxyl methyltransferase (Icmt) binding pocket: sulfonamide modified farnesyl cysteine (SMFC) analogs as Icmt inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters May 2011
- 2616-20 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1464-3405
10.1016/j.bmcl.2011.01.078 doi
Binding Sites
Cysteine--analogs & derivatives
Enzyme Activation--drug effects
Enzyme Inhibitors--chemistry
Humans
Inhibitory Concentration 50
Molecular Structure
Protein Methyltransferases--antagonists & inhibitors
Protein Processing, Post-Translational