HIV-1 integrase strand transfer inhibitors stabilize an integrase-single blunt-ended DNA complex. [electronic resource]
- Journal of molecular biology Jul 2011
- 831-46 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1089-8638
10.1016/j.jmb.2011.01.043 doi
Base Pairing--genetics Biocatalysis--drug effects Carbocyanines--metabolism DNA--metabolism DNA Footprinting Deoxyribonuclease I--metabolism Drug Resistance, Viral--drug effects Electrophoresis, Agar Gel Fluorescent Dyes--metabolism HIV Integrase--metabolism HIV Long Terminal Repeat--genetics HIV-1--drug effects Humans Inhibitory Concentration 50 Integrase Inhibitors--chemistry Keto Acids--chemistry Mutant Proteins--metabolism Protein Binding--drug effects Protein Multimerization--drug effects Pyrrolidinones--chemistry Raltegravir Potassium Substrate Specificity--drug effects