Genetic ablation of delta opioid receptors in nociceptive sensory neurons increases chronic pain and abolishes opioid analgesia. [electronic resource]
- Pain Jun 2011
- 1238-1248 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
1872-6623
10.1016/j.pain.2010.12.031 doi
Analgesics, Opioid--therapeutic use Analysis of Variance Animals Benzamides--therapeutic use Disease Models, Animal Dose-Response Relationship, Drug Freund's Adjuvant--adverse effects Ganglia, Spinal--pathology Guanosine 5'-O-(3-Thiotriphosphate)--pharmacokinetics Inflammation--chemically induced Mice Mice, Inbred C57BL Motor Activity--drug effects NAV1.8 Voltage-Gated Sodium Channel Nociceptors--drug effects Pain--etiology Pain Measurement--methods Piperazines--therapeutic use Protein Binding--drug effects Receptors, Opioid, delta--deficiency Sodium Channels--genetics Sulfur Isotopes--pharmacokinetics