Dowal, Louisa

Identification of an antithrombotic allosteric modulator that acts through helix 8 of PAR1. [electronic resource] - Proceedings of the National Academy of Sciences of the United States of America Feb 2011 - 2951-6 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1091-6490

10.1073/pnas.1014863108 doi


Allosteric Regulation--physiology
Animals
Antithrombins--metabolism
Calcium--metabolism
Cell Line
Dogs
Epinephrine
Flow Cytometry
Luciferases
P-Selectin--metabolism
Peptide Fragments--metabolism
Platelet Aggregation
Protein Structure, Secondary--physiology
Receptor, PAR-1--agonists
Receptors, G-Protein-Coupled--metabolism
Signal Transduction--physiology
Thrombosis--metabolism